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ActivX News Releases
03/21/07
ActivX Biosciences Launches Breakthrough Kinase Platform, KiNativ™
03/15/06
ActivX/Kyorin Begins First U.S. Phase I Study for Novel Anti-Diabetic Drug
03/14/06
ActivX Biosciences Announces Expansion of Strategic Collaboration Agreement with Pfizer Inc. with Multiple Discovery and Developmental Stage Projects
02/10/05
Wall Street Reporter Interview with Dr. John Kozarich
02/09/05
ActivX Biosciences Announces Expansion of Strategic Collaboration Agreement with Pfizer Inc. with Multiple Discovery and Developmental Stage Projects
02/03/05
BioWorld Today article on Kyorin purchase of ActivX Biosciences
02/02/05
ActivX Biosciences Announces Closing of Aquisition by Kyorin Pharmaceutical Co., Ltd.
Pre 2005 Press
ActivX Publications
01/2007
Polo-like kinases inhibited by wortmannin. Labeling site and downstream effects
01/2007
Synthesis and activity of a potent, specific azabicyclo[3.3.0]-octane-based DPP II inhibitor
01/2007
Functional Interrogation of the Kinome using Nucleotide Acyl Phosphates
10/2005
Boro-norleucine as a P1 residue for the design of selective and potent DPP7 inhibitorsent DPP7 inhibitors
10/2005
Synthesis and structure-activity relationship of N-alkyl Gly-boro-Pro inhibitors of DPP4, FAP, and DPP7
04/2005
Clinical Proteomics
02/2005
High-resolution functional proteomics by active-site peptide profiling
01/2005
Wortmannin, a Widely Used Phosphoinositide 3-Kinase Inhibitor, also Potently Inhibits Mammalian Polo-like Kinase
03/2004
Synergistic Computational and Experimental Proteomics Approaches for More Accurate Detection of Active Serine Hydrolases in Yeast
01/2004
Mapping Enzyme Active Sites in Complex Proteomes
08/2003
Prolyl peptidases: a serine protease subfamily with high potential for drug discovery
04/2003
Proteomic Tools for Quantitation by Mass Spectrometry
04/2003
Functional profiling of the proteome with affinity labels
02/2003
Activity-based proteomics: enzyme chemistry redux
02/2003
Inhibitor Focusing: Direct Selection of Drug Targets from Proteomes Using Activity-Based Probes
08/2002
Enzyme activity profiles of the secreted and membrane proteome that depict cancer cell invasiveness
07/2002
Activity-based probes for functional proteomics
09/2001
Direct visualization of serine hydrolase activities in complex proteomes using fluorescent active site-directed probes
03/2001
Profiling Serine Hydrolase Activities in Complex Proteomes
12/1999
Activity-based protein profiling: The serine hydrolases